SCHEMBL6957708

SCHEMBL6957708

N#Cc1ccc2[nH]cc(CCCCN3CCCC(Cc4ccccc4)C3)c2c1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.61
HTR1A P08908 8/20 0.56
ACHE P22303 1/20 0.56
SLC6A2 P23975 1/20 0.56
SLC6A3 Q01959 1/20 0.56
HTR6 P50406 1/20 0.54
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954897 1.00 SLC6A4 (0.61) SLC6A4HTR1AACHESLC6A2SLC6A3
SCHEMBL6954494 1.00 SLC6A4 (0.61) SLC6A4HTR1AACHESLC6A2SLC6A3
SCHEMBL6953432 0.93 SLC6A4 (0.52) SLC6A4HTR1AACHESLC6A2SLC6A3
SCHEMBL6958552 0.86 MPO (0.61) SLC6A4HTR1AKCNH2
SCHEMBL6951363 0.86 HTR1A (0.55) SLC6A4HTR1AHTR6KCNH2
SCHEMBL6952634 0.86 MPO (0.61) SLC6A4HTR1AKCNH2
SCHEMBL7358948 0.86 HTR1A (0.54) SLC6A4HTR1A
SCHEMBL6957729 0.86 MPO (0.61) SLC6A4HTR1AKCNH2
SCHEMBL6950516 0.86 HTR1A (0.56) SLC6A4HTR1AHTR6
SCHEMBL7384064 0.84 HTR1A (0.48) SLC6A4HTR1AACHESLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP disclosed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO disclosed