SCHEMBL6963779

SCHEMBL6963779

Cc1c(C(O)CCc2cn(C(c3ccccc3)(c3ccccc3)c3ccccc3)cn2)sc2ccc(F)cc12

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 15/20 0.39
NMBR P28336 1/20 0.33
HTR1A P08908 1/20 0.32
CRHR1 P34998 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963554 0.86 SIRT2 (0.38) SIRT2NMBR
SCHEMBL6960303 0.81 SIRT2 (0.39) SIRT2
SCHEMBL6958792 0.80 SIRT2 (0.38) SIRT2
SCHEMBL6964092 0.79 SIRT2 (0.38) SIRT2
SCHEMBL6952126 0.70 MAPT (0.36) SIRT2
SCHEMBL6952132 0.70 MAPT (0.36) SIRT2
SCHEMBL1037984 0.69 SIRT2 (0.40) SIRT2NMBR
SCHEMBL8979144 0.69 SIRT2 (0.42) SIRT2HTR1A
SCHEMBL7084465 0.69 SIRT2 (0.44) SIRT2HTR1A
SCHEMBL6958299 0.68 CYP19A1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed