SCHEMBL6960199

SCHEMBL6960199

COC(=O)c1ccc([N+](=O)[O-])cc1[N+](=O)[O-]

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.55
CES2 O00748 1/20 0.55
MAPT P10636 4/20 0.54
POLB P06746 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.51
ALDH1A1 P00352 3/20 0.51
MAPK1 P28482 2/20 0.51
TP53 P04637 1/20 0.51
HPGD P15428 1/20 0.51
TSHR P16473 1/20 0.51
GPR35 Q9HC97 1/20 0.51
HTT P42858 1/20 0.50
FLT1 P17948 1/20 0.50
FLT4 P35916 1/20 0.50
KDR P35968 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
LMNA P02545 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nornitrogen Mustard SCHEMBL8638765 0.88 KDM4E (0.49) KDM4ECES2MAPTPOLBSMN1; SMN2
SCHEMBL1403472 0.86 ALDH1A1 (0.56) KDM4EMAPTPOLBSMN1; SMN2ALDH1A1
SCHEMBL9502855 0.86 CES2 (0.58) KDM4ECES2MAPTPOLBSMN1; SMN2
SCHEMBL11130755 0.86 CES2 (0.58) KDM4ECES2MAPTPOLBSMN1; SMN2
SCHEMBL30203403 0.86 ALDH1A1 (0.56) KDM4EMAPTPOLBSMN1; SMN2ALDH1A1
Methane SCHEMBL27588822 0.85 ALDH1A1 (0.54) KDM4EMAPTPOLBSMN1; SMN2ALDH1A1
SCHEMBL11169142 0.85 CES2 (0.56) KDM4ECES2MAPTPOLBSMN1; SMN2
SCHEMBL30179515 0.85 CES2 (0.56) KDM4ECES2MAPTPOLBSMN1; SMN2
SCHEMBL23037541 0.83 CES2 (0.55) KDM4ECES2MAPTPOLBSMN1; SMN2
SCHEMBL559830 0.83 VCAM1 (0.64) KDM4EMAPTPOLBSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110713454-A Nitro-substituted indole compound and preparation method thereof 南京工业大学 2020-01-21 CN claimed
CN-110713454-A Nitro-substituted indole compound and preparation method thereof 南京工业大学 2020-01-21 CN disclosed
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed
US-4054556-A Polyurethanes cured with derivatives of 2,4-diamino-benzoic acid E. I. DU PONT DE NEMOURS AND COMPANY (US) 1977-10-18 US disclosed
US-4039514-A SUBSTITUTED 2,4-DIAMINOBENZOIC ACID E. I. DU PONT DE NEMOURS AND COMPANY (US) 1977-08-02 US disclosed