SCHEMBL6960591

SCHEMBL6960591

CC(C)c1nc(CN=C(N)N)n(Cc2ccncc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
KCNH2 Q12809 1/20 0.33
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
HSP90B1 P14625 1/20 0.32
TRAP1 Q12931 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084720 0.91 HTR3E (0.40) PIM1PIM3KCNH2HTR3EHTR3B
SCHEMBL7078779 0.89 ADRA1D (0.35) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL6966455 0.89 PIM1 (0.31) PIM1PIM3
SCHEMBL6967507 0.88 PIM1 (0.34) PIM1PIM3TDP1MEN1KMT2A
SCHEMBL5852651 0.87 KCNH2 (0.35) PIM1PIM3KCNH2HSP90B1TRAP1
SCHEMBL6957548 0.87 KCNH2 (0.35) PIM1PIM3KCNH2HSP90B1TRAP1
SCHEMBL14439807 0.86 KCNH2 (0.38) KCNH2HSP90B1TRAP1TDP1MEN1
SCHEMBL6969033 0.86 HSP90B1 (0.32) HTR3EHTR3BHTR3AHTR3DHTR3C
Carbamic Acid SCHEMBL667612 0.86 PIM1 (0.36) PIM1PIM3KCNH2HSP90B1TRAP1
SCHEMBL6967022 0.85 ADRA1D (0.34) HSP90B1TRAP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed