SCHEMBL6967022

SCHEMBL6967022

CC(C)c1nc(CN=C(N)N)n(Cc2ccccn2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.34
HSP90B1 P14625 1/20 0.31
TRAP1 Q12931 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
S1PR3 Q99500 1/20 0.31
ALDH1A1 P00352 1/20 0.31
AGTR1 P30556 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
TP53 P04637 1/20 0.31
XIAP P98170 1/20 0.31
BIRC2 Q13490 1/20 0.31
GRIN2D O15399 1/20 0.30
GRIN3B O60391 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2B Q13224 1/20 0.30
GRIN2C Q14957 1/20 0.30
GRIN3A Q8TCU5 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957969 0.93 HTR3E (0.35) ADRA1DALDH1A1AGTR1HRH4TP53
SCHEMBL6973295 0.89 HRH4 (0.34) TLR7ALDH1A1HRH4TP53GRIN2D
SCHEMBL6973165 0.89 S1PR3 (0.34) TLR7S1PR3ALDH1A1HRH4GRIN2D
SCHEMBL6976953 0.88 ALDH1A1 (0.33) ADRA1DHSP90B1TRAP1TLR7S1PR3
SCHEMBL6975001 0.88 ALDH1A1 (0.33) ADRA1DHSP90B1TRAP1TLR7ALDH1A1
SCHEMBL7082531 0.86 HRH1 (0.34) ADRA1DHSP90B1TRAP1TLR7S1PR3
SCHEMBL7082928 0.86 HRH1 (0.36) ADRA1DHSP90B1TRAP1TLR7S1PR3
SCHEMBL6960591 0.85 PIM1 (0.33) HSP90B1TRAP1MEN1KMT2A
SCHEMBL6962934 0.85 MEN1 (0.39) ADRA1DS1PR3ALDH1A1TP53XIAP
SCHEMBL7078156 0.85 GRIN1 (0.36) S1PR3ALDH1A1HRH4GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed