SCHEMBL6961647

SCHEMBL6961647

O=[N+]([O-])c1ccc(Sc2cccc3cnccc23)cc1NCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
HTR6 P50406 4/20 0.44
POLB P06746 2/20 0.44
MAPT P10636 6/20 0.44
NPSR1 Q6W5P4 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PKM P14618 2/20 0.43
LMNA P02545 1/20 0.43
APP P05067 2/20 0.43
ALDH1A1 P00352 2/20 0.42
GAA P10253 2/20 0.42
HTT P42858 2/20 0.42
SIRT6 Q8N6T7 1/20 0.42
USP2 O75604 1/20 0.41
RECQL P46063 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966199 0.83 HDAC6 (0.42) MEN1KMT2AMAPTCYP1A2CYP3A4
SCHEMBL6966909 0.78 KDM4E (0.43) MEN1KMT2AMAPTNPSR1LMNA
SCHEMBL6966094 0.78 LMNA (0.43) MEN1KMT2AMAPTNPSR1CYP1A2
SCHEMBL6967573 0.76 HTT (0.47) MEN1KMT2APOLBMAPTNPSR1
SCHEMBL8567878 0.74 KDM4C (0.57) MEN1KMT2AHTR6POLBMAPT
SCHEMBL6963693 0.73 MAPT (0.60) MEN1KMT2APOLBMAPTNPSR1
SCHEMBL432366 0.72 HTR6 (0.61) HTR6POLBMAPTNPSR1PKM
SCHEMBL6972315 0.71 LMNA (0.46) MEN1KMT2APOLBMAPTNPSR1
SCHEMBL12205175 0.71 HTR6 (0.66) MEN1KMT2AHTR6MAPTNPSR1
SCHEMBL8664733 0.71 ALDH1A1 (0.62) MEN1KMT2AHTR6POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed