SCHEMBL6962273

SCHEMBL6962273

CCOC(=O)C1=C(c2ccc(F)cc2)NC(C)=C(C(=O)OC)C1C(C)C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.58
CACNA1F O60840 1/20 0.52
CACNA1D Q01668 1/20 0.52
CACNA1S Q13698 1/20 0.52
CACNA1C Q13936 1/20 0.52
ALDH1A1 P00352 2/20 0.45
TRPV1 Q8NER1 2/20 0.45
KDM4E B2RXH2 4/20 0.45
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA7 P43166 2/20 0.45
CA9 Q16790 2/20 0.45
EPHX2 P34913 1/20 0.43
TMIGD3 P0DMS9 1/20 0.43
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962850 0.82 ALDH1A1 (0.50) ADORA3CACNA1CALDH1A1KDM4ECA12
SCHEMBL8193038 0.77 CACNA1F (0.57) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9272237 0.76 ADORA3 (0.39) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9263843 0.75 CA12 (0.47) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7687307 0.74 ADORA3 (1.00) ADORA3CACNA1DALDH1A1TRPV1TMIGD3
SCHEMBL2648819 0.73 CACNA1F (0.70) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL6961962 0.72 ALDH1A1 (0.48) ADORA3CACNA1CALDH1A1KDM4ECA12
SCHEMBL10297381 0.71 SMN1; SMN2 (0.45) ADORA3CACNA1CALDH1A1KDM4ECA12
SCHEMBL9831380 0.68 KDM4E (0.86) ADORA3ALDH1A1KDM4EMEN1CYP1A2
SCHEMBL8106730 0.68 KDM4E (0.86) ADORA3ALDH1A1KDM4EMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325130-B1 Substituted pyridines BAYER AG (DE) 2003-11-05 EP disclosed
EP-1123925-A1 Process for preparation of substituted pyridines BAYER AG (DE) 2001-08-16 EP disclosed
EP-1123924-A1 Substituted pyridines as HMG-COA reductase inhibitors BAYER AG (DE) 2001-08-16 EP disclosed
US-5401746-A FOR INHIBITING CHOLESTEROL BIOSYNTHESIS AND HMG-COA REDUCTASE BAYER AKTIENGESELLSCHAFT (DE) 1995-03-28 US disclosed
US-5169857-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1992-12-08 US disclosed
US-5006530-A Certain 7-[2,6-diisopropyl-4-phenyl-5-lower alkoxymethyl-pyrid-3-yl]-3,5-dihydroxy-6-enoates and derivatives useful for treating circulatory diseases BAYER AKTIENGESELLSCHAFT (DE) 1991-04-09 US disclosed
EP-0325130-A2 Substituted pyridines BAYER AG (DE) 1989-07-26 EP disclosed