SCHEMBL6962276

SCHEMBL6962276

N=C(Nc1ccc(CCNCc2ccc(Cl)cc2)cc1)c1cccs1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.52
RAB9A P51151 4/20 0.52
MAPT P10636 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
NOS3 P29474 3/20 0.49
NOS1 P29475 2/20 0.49
NOS2 P35228 2/20 0.49
POLB P06746 2/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
HTT P42858 1/20 0.48
CNR1 P21554 5/20 0.45
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
BCHE P06276 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958210 0.90 GAA (0.49) NPC1RAB9AMAPTSMN1; SMN2NOS3
SCHEMBL6963560 0.90 GAA (0.49) NPC1RAB9AMAPTSMN1; SMN2NOS3
SCHEMBL29558856 0.89 NOS3 (0.64) NPC1RAB9AMAPTSMN1; SMN2NOS3
SCHEMBL122445 0.89 NOS3 (0.64) NPC1RAB9AMAPTSMN1; SMN2NOS3
SCHEMBL27357975 0.88 NOS3 (0.47) NPC1RAB9AMAPTSMN1; SMN2NOS3
SCHEMBL4397478 0.88 ALDH1A1 (0.44) SMN1; SMN2NOS3NOS1NOS2KDM4E
SCHEMBL9039601 0.88 NPC1 (0.48) NPC1RAB9AMAPTSMN1; SMN2NOS3
Hydrochloric Acid SCHEMBL31114391 0.88 NOS3 (0.65) NPC1RAB9AMAPTSMN1; SMN2NOS3
SCHEMBL6962883 0.87 NOS3 (0.49) NPC1RAB9AMAPTSMN1; SMN2NOS3
Hydrochloric Acid SCHEMBL6962460 0.87 NPC1 (0.47) NPC1RAB9AMAPTSMN1; SMN2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP claimed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO claimed
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed