SCHEMBL6962883

SCHEMBL6962883

N=C(Nc1ccc(CCNCc2ccc(Cl)c(Cl)c2)cc1)c1cccs1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.49
NOS1 P29475 2/20 0.49
NOS2 P35228 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
MAPT P10636 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
F7 P08709 1/20 0.39
NR1I3 Q14994 1/20 0.39
LMNA P02545 2/20 0.39
KMT2A Q03164 2/20 0.39
ROCK1 Q13464 1/20 0.39
HSP90AA1 P07900 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29558856 0.88 NOS3 (0.64) NOS3NOS1NOS2CYP1A2CYP2D6
SCHEMBL122445 0.88 NOS3 (0.64) NOS3NOS1NOS2CYP1A2CYP2D6
SCHEMBL6962276 0.87 NPC1 (0.52) NOS3NOS1NOS2MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL31114391 0.87 NOS3 (0.65) NOS3NOS1NOS2CYP1A2CYP2D6
SCHEMBL15499648 0.86 NOS3 (0.51) NOS3NOS1NOS2CYP1A2CYP2D6
SCHEMBL6967375 0.86 NOS3 (0.46) NOS3NOS1NOS2MAPTSMN1; SMN2
SCHEMBL6964306 0.85 NOS3 (0.43) NOS3NOS1NOS2CYP2D6CYP2C9
SCHEMBL6958210 0.85 GAA (0.49) NOS3NOS1NOS2CYP1A2CYP2C9
SCHEMBL6963560 0.85 GAA (0.49) NOS3NOS1NOS2CYP1A2CYP2C9
SCHEMBL6961265 0.83 NOS1 (0.48) NOS3NOS1NOS2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP claimed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO claimed
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed