SCHEMBL6962571

SCHEMBL6962571

CC(=O)OCCOC(Cc1cccnc1)c1nc(C(C)C)c(Sc2cccc([N+](=O)[O-])c2)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.36
FKBP1A P62942 1/20 0.35
CYP19A1 P11511 3/20 0.34
CYP11B1 P15538 3/20 0.34
CYP11B2 P19099 3/20 0.34
ATM Q13315 1/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 3/20 0.33
MAPT P10636 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP2C19 P33261 3/20 0.33
CYP2D6 P10635 2/20 0.33
RECQL P46063 1/20 0.33
MEN1 O00255 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
KMT2A Q03164 2/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
THPO P40225 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967395 0.92 MEN1 (0.35) RXFP1ATMALDH1A1LMNAMAPT
SCHEMBL6974934 0.91 CYP19A1 (0.35) RXFP1FKBP1ACYP19A1CYP11B1CYP11B2
SCHEMBL6972999 0.91 RXFP1 (0.37) RXFP1FKBP1ACYP19A1CYP11B1CYP11B2
SCHEMBL6960778 0.88 LMNA (0.34) ALDH1A1LMNAMAPTMEN1CYP1A2
SCHEMBL7084647 0.88 ALDH1A1 (0.38) ALDH1A1LMNAMEN1KMT2AKDM4E
SCHEMBL6973132 0.88 LMNA (0.34) LMNARECQLMEN1CYP1A2CYP3A4
SCHEMBL6971934 0.87 CACNA1C (0.35) ATMLMNAMAPTCYP2C9CYP2C19
SCHEMBL6975428 0.86 CYP1A2 (0.35) ALDH1A1LMNAMAPTCYP2C9CYP2C19
SCHEMBL7082209 0.85 IDO1 (0.34) MEN1CYP1A2CYP3A4KMT2AKDM4E
SCHEMBL6969216 0.85 MEN1 (0.34) ALDH1A1LMNAMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed