SCHEMBL6975428

SCHEMBL6975428

CC(=O)OCCOC(Cc1ccccn1)c1nc(C(C)C)c(Sc2cccc([N+](=O)[O-])c2)[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.35
CYP3A4 P08684 3/20 0.35
MEN1 O00255 6/20 0.35
KMT2A Q03164 6/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
ALDH1A1 P00352 5/20 0.33
KDM4E B2RXH2 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
MAPT P10636 2/20 0.32
MAPK1 P28482 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
PKM P14618 1/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
LMNA P02545 2/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
THPO P40225 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969928 0.91 CYP1A2 (0.35) CYP1A2CYP3A4MEN1KMT2ANPC1
SCHEMBL7084594 0.90 CYP1A2 (0.38) CYP1A2CYP3A4MEN1KMT2ANPC1
SCHEMBL7080029 0.88 PTPRA (0.34) CYP1A2NPC1ALDH1A1MAPTSMN1; SMN2
SCHEMBL6967395 0.88 MEN1 (0.35) CYP1A2CYP3A4MEN1KMT2AALDH1A1
SCHEMBL7078551 0.88 SLC6A9 (0.33) KMT2A
SCHEMBL6973420 0.88 SMN1; SMN2 (0.35) KMT2ANPC1RAB9AALDH1A1MAPT
SCHEMBL6971934 0.88 CACNA1C (0.35) CYP1A2CYP3A4MEN1KMT2AMAPT
SCHEMBL6962571 0.86 RXFP1 (0.36) CYP1A2CYP3A4MEN1KMT2ARAB9A
SCHEMBL7085474 0.85 CYP2C9 (0.38) CYP1A2CYP3A4MEN1KMT2ANPC1
SCHEMBL8113590 0.84 MAOB (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed