SCHEMBL6963230

SCHEMBL6963230

Cn1nccc1-c1ccc2c(ccn2-c2ccc(F)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.53
KCNH2 Q12809 1/20 0.51
HTR1A P08908 1/20 0.44
HTR1B P28222 1/20 0.44
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PI4KA P42356 1/20 0.40
PIK3CG P48736 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
NT5E P21589 2/20 0.39
NR3C1 P04150 5/20 0.38
FAAH O00519 1/20 0.38
PGR P06401 3/20 0.38
AXL P30530 1/20 0.37
MAOB P27338 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967276 0.77 DRD2 (0.55) DRD2KCNH2HTR1AHTR1BPIK3CA
SCHEMBL6957221 0.77 KCNH2 (0.51) KCNH2HTR1AHTR1BNR3C1FAAH
SCHEMBL6957036 0.77 KCNH2 (0.54) DRD2KCNH2NR3C1PGRMAPT
SCHEMBL6964471 0.76 DRD2 (0.54) DRD2KCNH2HTR1AHTR1BPIK3CD
SCHEMBL6967960 0.76 KCNH2 (0.50) DRD2KCNH2HTR1AHTR1BNR3C1
SCHEMBL6966467 0.76 KCNH2 (0.52) KCNH2HTR1AHTR1BNR3C1FAAH
SCHEMBL3489735 0.75 CYP1A2 (0.53) DRD2KCNH2PIK3CDPIK3CAPIK3CB
SCHEMBL6960229 0.74 DRD2 (0.54) DRD2KCNH2HTR1AHTR1BFAAH
SCHEMBL6966566 0.73 KCNH2 (0.50) DRD2KCNH2HTR1AHTR1BMAOB
SCHEMBL6961517 0.73 DRD2 (0.54) DRD2KCNH2HTR1AHTR1BNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602889-B1 5-heteroaryl substituted indoles H. LUNDBECK A.S. (DK) 2003-08-05 US disclosed
EP-1068198-B1 5-HETEROARYL SUBSTITUTED INDOLES LUNDBECK & CO AS H (DK) 2003-05-28 EP disclosed