SCHEMBL6967960

SCHEMBL6967960

Cn1ncc(-c2ccc3c(ccn3-c3ccc(F)cc3)c2)n1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.50
HTR1A P08908 2/20 0.44
HTR1B P28222 2/20 0.44
NR3C1 P04150 9/20 0.40
DRD2 P14416 3/20 0.39
PGR P06401 5/20 0.39
MCHR1 Q99705 1/20 0.36
MAOB P27338 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
FAAH O00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6965840 0.85 KCNH2 (0.48) KCNH2HTR1AHTR1BNR3C1DRD2
SCHEMBL6964471 0.83 DRD2 (0.54) KCNH2HTR1AHTR1BNR3C1DRD2
SCHEMBL6960229 0.79 DRD2 (0.54) KCNH2HTR1AHTR1BDRD2MAOB
SCHEMBL6967276 0.79 DRD2 (0.55) KCNH2HTR1AHTR1BNR3C1DRD2
SCHEMBL6966566 0.78 KCNH2 (0.50) KCNH2HTR1AHTR1BDRD2MAOB
SCHEMBL6963230 0.76 DRD2 (0.53) KCNH2HTR1AHTR1BNR3C1DRD2
SCHEMBL5047902 0.76 AOC3 (0.47) HTR1AHTR1BMEN1NPC1ALDH1A1
SCHEMBL6961517 0.75 DRD2 (0.54) KCNH2HTR1AHTR1BNR3C1DRD2
SCHEMBL6966311 0.75 KCNH2 (0.52) KCNH2HTR1AHTR1BNR3C1DRD2
SCHEMBL6960921 0.74 KCNH2 (0.49) KCNH2NR3C1KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602889-B1 5-heteroaryl substituted indoles H. LUNDBECK A.S. (DK) 2003-08-05 US disclosed
EP-1068198-B1 5-HETEROARYL SUBSTITUTED INDOLES LUNDBECK & CO AS H (DK) 2003-05-28 EP disclosed