SCHEMBL6963265

SCHEMBL6963265

N#Cc1ccc(Sc2cccc3cnccc23)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.47
SLC22A12 Q96S37 3/20 0.39
CHUK O15111 1/20 0.39
CYP3A4 P08684 2/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
ROCK2 O75116 2/20 0.37
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
CYP17A1 P05093 1/20 0.36
CYP3A5 P20815 1/20 0.36
AR P10275 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963171 0.85 AR (0.53) HTTSLC22A12CHUKCYP3A4KDM4E
SCHEMBL6961639 0.80 MAPT (0.45) HTTSLC22A12KDM4ELMNAALDH1A1
SCHEMBL6968741 0.78 KDM4E (0.57) HTTSLC22A12CYP3A4KDM4ELMNA
SCHEMBL6973379 0.76 CYP3A4 (0.51) HTTCYP3A4KDM4ELMNACYP1A2
SCHEMBL6967708 0.73 HTT (0.45) HTTSLC22A12CHUKCYP3A4KDM4E
SCHEMBL6973375 0.70 LMNA (0.54) HTTCYP3A4KDM4ELMNACYP1A2
SCHEMBL6962431 0.69 HTT (0.52) HTTSLC22A12CYP3A4KDM4ELMNA
SCHEMBL6958271 0.68 LMNA (0.42) HTTCYP3A4KDM4ELMNACYP1A2
SCHEMBL25625881 0.68 CYP11B2 (0.50) HTTSLC22A12CHUKCYP11B1CYP11B2
SCHEMBL4207818 0.66 KDM4E (0.59) HTTCYP3A4KDM4ELMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed