SCHEMBL6963360

SCHEMBL6963360

O=c1oc(-c2ccc(OCc3ccncc3)cc2)cc(O)c1SCCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.46
ABCB1 P08183 1/20 0.45
MAPT P10636 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
PTPN1 P18031 4/20 0.43
NPC1 O15118 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PRKDC P78527 1/20 0.42
SMPD1 P17405 1/20 0.41
GSTP1 P09211 1/20 0.41
F2 P00734 1/20 0.41
KCNH2 Q12809 1/20 0.41
GRIN2B Q13224 1/20 0.41
MCL1 Q07820 1/20 0.41
ACHE P22303 1/20 0.40
MAOB P27338 1/20 0.40
TERT O14746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6952547 0.94 ABCB1 (0.50) ABCB1MAPTL3MBTL1PTPN1PRKDC
SCHEMBL6963290 0.91 TERT (0.43) ABCB1MAPTL3MBTL1PTPN1HTT
SCHEMBL6950945 0.88 GSK3B (0.47) L3MBTL1NPC1HTTSMN1; SMN2
SCHEMBL6965573 0.87 ABCB1 (0.40) ABCB1MAPTL3MBTL1PTPN1SMN1; SMN2
SCHEMBL6954678 0.86 ABCB1 (0.43) ABCB1MAPTL3MBTL1NPC1PRKDC
SCHEMBL6956331 0.86 SLC16A3 (0.46) ABCB1MAPTL3MBTL1NPC1PRKDC
SCHEMBL6958378 0.85 MAOA (0.45) ABCB1ACHEMAOB
SCHEMBL6960907 0.85 ACHE (0.42) ABCB1MAPTL3MBTL1SMN1; SMN2ACHE
SCHEMBL6953671 0.85 MRGPRX4 (0.48) SMN1; SMN2
SCHEMBL6952541 0.85 MAOB (0.45) ABCB1MAPTL3MBTL1PRKDCKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5808062-A AIDS THERAPY WARNER-LAMBERT COMPANY (US) 1998-09-15 US claimed
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP claimed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO claimed
EP-0729465-B1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2003-01-22 EP disclosed
US-6005103-A TREATMENT OF BACTERIAL AND VIRAL INFECTIONS AND DISEASES, INCLUDING AIDS WARNER-LAMBERT COMPANY (US) 1999-12-21 US disclosed
US-5808062-A AIDS THERAPY WARNER-LAMBERT COMPANY (US) 1998-09-15 US disclosed
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
EP-0729465-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014013-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed