SCHEMBL6963909

SCHEMBL6963909

Cc1nc(Nc2ccc(F)cc2)nc(N2CCc3cc(OC(=O)C(COCc4ccccc4)NC(=O)OC(C)(C)C)ccc3C2C)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 2/20 0.40
KLK5 Q9Y337 2/20 0.40
PPARA Q07869 2/20 0.38
CTSS P25774 1/20 0.37
P2RX7 Q99572 1/20 0.36
PABPC1 P11940 1/20 0.35
PPARG P37231 1/20 0.35
GHSR Q92847 4/20 0.35
CCKBR P32239 1/20 0.35
UGCG Q16739 2/20 0.34
RAB9A P51151 1/20 0.34
PTPN1 P18031 3/20 0.34
CDC25B P30305 3/20 0.34
PTPN2 P17706 2/20 0.34
CDC25A P30304 1/20 0.34
CCNT1 O60563 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CDK9 P50750 1/20 0.34
CCNA1 P78396 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963911 1.00 KLK7 (0.40) KLK7KLK5PPARACTSSP2RX7
SCHEMBL6957715 0.95 KLK7 (0.40) KLK7KLK5PPARACTSSP2RX7
SCHEMBL6957710 0.95 KLK7 (0.40) KLK7KLK5PPARACTSSP2RX7
SCHEMBL6965676 0.93 PABPC1 (0.41) CTSSP2RX7PABPC1SCN9A
SCHEMBL6965678 0.93 PABPC1 (0.41) CTSSP2RX7PABPC1SCN9A
SCHEMBL6968593 0.89 SCN9A (0.33) P2RX7PABPC1GHSRSCN9A
SCHEMBL6963915 0.89 SCN9A (0.36) P2RX7PABPC1GHSRSCN9A
SCHEMBL6967714 0.88 PABPC1 (0.41) CTSSP2RX7PABPC1SCN9A
SCHEMBL6967718 0.88 PABPC1 (0.41) CTSSP2RX7PABPC1SCN9A
SCHEMBL6963190 0.88 SCN9A (0.39) PABPC1GHSRSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015444-B1 PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP LTD (KR) 2003-05-28 EP disclosed