SCHEMBL6964366

SCHEMBL6964366

CC(c1c[nH]c2ccc(C3CCOCC3)cc12)C1CCCN1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.38
TLR9 Q9NR96 13/20 0.36
TLR8 Q9NR97 13/20 0.36
TLR7 Q9NYK1 13/20 0.36
PRKAB2 O43741 2/20 0.34
PRKAG1 P54619 2/20 0.34
PRKAA2 P54646 2/20 0.34
PRKAA1 Q13131 2/20 0.34
PRKAG3 Q9UGI9 2/20 0.34
PRKAG2 Q9UGJ0 2/20 0.34
PRKAB1 Q9Y478 2/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
MAPK1 P28482 1/20 0.33
SOS1 Q07889 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962926 0.90 HTR1D (0.47) HTR1DTLR9TLR8TLR7SLC6A2
SCHEMBL6974690 0.89 TLR9 (0.41) HTR1DTLR9TLR8TLR7
SCHEMBL6976838 0.83 PRKAG1 (0.38) HTR1DPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL25340081 0.82 TLR9 (0.43) HTR1DTLR9TLR8TLR7PRKAB2
SCHEMBL6960603 0.82 HTR1D (0.36) HTR1DTLR9TLR8TLR7SLC6A2
SCHEMBL8507358 0.81 HTR1D (0.45) HTR1DSLC6A2SLC6A4SLC6A3
SCHEMBL6971259 0.81 SLC6A2 (0.32) SLC6A2SLC6A4SLC6A3
SCHEMBL8208352 0.80 HTR1D (0.40) HTR1DSLC6A2SLC6A4SLC6A3
SCHEMBL6970050 0.80 SLC6A2 (0.32) SLC6A2SLC6A4SLC6A3
SCHEMBL6975409 0.79 SLC6A2 (0.32) HTR1DSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP claimed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed