SCHEMBL6962926

SCHEMBL6962926

CC(c1c[nH]c2ccc(C3CCCCC3)cc12)C1CCCN1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.47
SLC6A4 P31645 4/20 0.39
SLC6A2 P23975 3/20 0.39
SLC6A3 Q01959 3/20 0.39
MEN1 O00255 2/20 0.34
TP53 P04637 2/20 0.34
MAPT P10636 2/20 0.34
MAPK1 P28482 2/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 1/20 0.34
CCR6 P51684 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974690 0.92 TLR9 (0.41) HTR1DTLR9TLR8TLR7
SCHEMBL6964366 0.90 HTR1D (0.38) HTR1DSLC6A4SLC6A2SLC6A3MAPK1
SCHEMBL6960603 0.87 HTR1D (0.36) HTR1DSLC6A4SLC6A2SLC6A3TLR9
SCHEMBL8507358 0.84 HTR1D (0.45) HTR1DSLC6A4SLC6A2SLC6A3HTR6
SCHEMBL6976838 0.83 PRKAG1 (0.38) HTR1DSLC6A4SLC6A2SLC6A3
SCHEMBL8208352 0.83 HTR1D (0.40) HTR1DSLC6A4SLC6A2SLC6A3TP53
SCHEMBL8209090 0.81 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3
SCHEMBL8209129 0.81 SLC6A4 (0.43) SLC6A4SLC6A2SLC6A3MAPK1KMT2A
SCHEMBL1697454 0.81 SLC6A4 (0.43) SLC6A4SLC6A2SLC6A3MEN1MAPT
SCHEMBL9287655 0.81 HTR1D (0.42) HTR1DSLC6A4SLC6A2SLC6A3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed