SCHEMBL6976838

SCHEMBL6976838

CC(c1c[nH]c2ccc(C3CCCCO3)cc12)C1CCCN1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PRKAG1 P54619 10/20 0.38
PRKAA1 Q13131 10/20 0.38
PRKAB1 Q9Y478 10/20 0.38
PRKAA2 P54646 9/20 0.38
PRKAB2 O43741 8/20 0.38
PRKAG3 Q9UGI9 8/20 0.38
PRKAG2 Q9UGJ0 8/20 0.38
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KDR P35968 4/20 0.33
TEK Q02763 4/20 0.33
HTR1D P28221 2/20 0.32
SLC6A9 P48067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962926 0.83 HTR1D (0.47) SLC6A2SLC6A4SLC6A3HTR1D
SCHEMBL6964366 0.83 HTR1D (0.38) PRKAG1PRKAA1PRKAB1PRKAA2PRKAB2
SCHEMBL6970050 0.82 SLC6A2 (0.32) SLC6A2SLC6A4SLC6A3
SCHEMBL6974690 0.80 TLR9 (0.41) HTR1D
SCHEMBL8507358 0.79 HTR1D (0.45) SLC6A2SLC6A4SLC6A3HTR1D
SCHEMBL6971259 0.79 SLC6A2 (0.32) SLC6A2SLC6A4SLC6A3
SCHEMBL8208352 0.78 HTR1D (0.40) SLC6A2SLC6A4SLC6A3HTR1D
SCHEMBL9287655 0.77 HTR1D (0.42) SLC6A2SLC6A4SLC6A3HTR1D
SCHEMBL774639 0.77 SLC6A4 (0.43) SLC6A2SLC6A4SLC6A3
SCHEMBL8209129 0.77 SLC6A4 (0.43) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP claimed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed