SCHEMBL6965305

SCHEMBL6965305

CC(=O)c1ccc(OS(=O)(=O)C(F)(F)F)c(C#N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
HSD11B1 P28845 1/20 0.40
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
AR P10275 1/20 0.37
PLA2G7 Q13093 3/20 0.37
ABCC9 O60706 2/20 0.37
ABCC8 Q09428 2/20 0.37
KCNJ11 Q14654 2/20 0.37
KCNJ8 Q15842 2/20 0.37
EPAS1 Q99814 3/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
GLA P06280 1/20 0.36
CYP3A4 P08684 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3909726 0.89 ALDH1A1 (0.51) ALDH1A1HPGDARPLA2G7EPAS1
SCHEMBL402630 0.87 NOTUM (0.43) ALDH1A1HPGDCYP11B1CYP11B2PLA2G7
SCHEMBL338554 0.84 SMN1; SMN2 (0.46) ALDH1A1HPGDKDM4EMAPT
SCHEMBL8326418 0.81 NOTUM (0.43) ALDH1A1HPGDCYP11B1CYP11B2AR
SCHEMBL7133735 0.80 ALDH1A1 (0.44) ALDH1A1HPGDCYP11B1CYP11B2AR
SCHEMBL1473470 0.80 HSD11B1 (0.40) ALDH1A1HSD11B1MAPT
SCHEMBL6314588 0.80 LMNA (0.47) ALDH1A1HSD11B1GAA
SCHEMBL2259279 0.80 AR (0.44) ARPLA2G7EPAS1
SCHEMBL8142488 0.79 NOTUM (0.46) ALDH1A1HPGDARKDM4EGAA
SCHEMBL881308 0.79 CA12 (0.50) ALDH1A1CYP1A2CYP3A4MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005070916-A1 THIOPHENE AND FURAN COMPOUNDS ELI LILLY AND COMPANY (US) 2005-08-04 WO disclosed
US-6649636-B1 Cyclooxygenase inhibitors PFIZER INC. 2003-11-18 US disclosed
EP-1104759-B1 Heteroaryl phenyl pyrazole compounds as anti-inflammatory/analgesic agents PFIZER PROD INC (US) 2003-10-22 EP disclosed
EP-1104759-A1 Heteroaryl phenyl pyrazole compounds as anti-inflammatory/analgesic agents Pfizer Products Inc. (US) 2001-06-06 EP disclosed