SCHEMBL6965501

SCHEMBL6965501

CCn1c(COCCOC(N)=O)nc(C(C)C)c1Sc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
ATM Q13315 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 2/20 0.31
TOP2A P11388 1/20 0.31
TOP2B Q02880 1/20 0.31
MAPT P10636 2/20 0.30
NPSR1 Q6W5P4 1/20 0.30
POLB P06746 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
TLR8 Q9NR97 1/20 0.30
TLR7 Q9NYK1 1/20 0.30
CXCL12 P48061 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086333 0.91 CYP1A2 (0.39) TSHRATMMEN1CYP1A2CYP2C9
SCHEMBL7081165 0.91 LMNA (0.35) LMNATSHRATMSMN1; SMN2MEN1
SCHEMBL7084632 0.91 SMN1; SMN2 (0.36) TSHRATMSMN1; SMN2MEN1CYP1A2
SCHEMBL6968991 0.89 LMNA (0.41) LMNATSHRATMMEN1CYP1A2
SCHEMBL7081807 0.89 ALOX12 (0.35) LMNASMN1; SMN2TP53
SCHEMBL7087212 0.89 EPHX1 (0.33) LMNAMEN1KMT2AALDH1A1MAPT
SCHEMBL6960266 0.88 CYP1A2 (0.36) LMNASMN1; SMN2MEN1CYP1A2CYP2C9
SCHEMBL7084824 0.87 PIM1 (0.34) LMNATSHRSMN1; SMN2MEN1CYP1A2
SCHEMBL6965379 0.86 CYP2C9 (0.36) LMNATSHRSMN1; SMN2MEN1CYP1A2
SCHEMBL6961556 0.86

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed