SCHEMBL7081165

SCHEMBL7081165

CCn1c(CCOC(N)=O)nc(C(C)C)c1Sc1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
ATM Q13315 1/20 0.35
CYP1A2 P05177 2/20 0.32
MEN1 O00255 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 2/20 0.32
CXCL12 P48061 1/20 0.32
POLB P06746 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
TP53 P04637 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 4/20 0.31
EPHX1 P07099 1/20 0.31
RECQL P46063 1/20 0.31
CYP2D6 P10635 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6968991 0.94 LMNA (0.41) LMNATSHRATMCYP1A2MEN1
SCHEMBL6965501 0.91 LMNA (0.33) LMNATSHRATMCYP1A2MEN1
SCHEMBL8116257 0.90 MEN1 (0.39) LMNATSHRATMCYP1A2MEN1
SCHEMBL7084632 0.89 SMN1; SMN2 (0.36) TSHRATMCYP1A2MEN1CYP2C9
SCHEMBL6975636 0.88 ALOX12 (0.36) LMNATP53
SCHEMBL6973633 0.88 EPHX1 (0.34) LMNAMEN1KMT2AALDH1A1MAPT
SCHEMBL8100016 0.87 LMNA (0.36) LMNACYP1A2MEN1CYP2C9CYP2C19
SCHEMBL6969118 0.86
SCHEMBL6968774 0.86 PIM1 (0.35) LMNACYP1A2MEN1CYP2C9CYP2C19
SCHEMBL7077278 0.85

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed