SCHEMBL7084632

SCHEMBL7084632

CCn1c(COC(N)=O)nc(C(C)C)c1Sc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.36
TSHR P16473 1/20 0.36
ATM Q13315 1/20 0.36
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP1A2 P05177 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TOP2A P11388 2/20 0.35
TOP2B Q02880 2/20 0.35
EPHX1 P07099 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CXCL12 P48061 1/20 0.33
MAPT P10636 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
CYP2D6 P10635 2/20 0.32
POLB P06746 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6965501 0.91 LMNA (0.33) SMN1; SMN2TSHRATMCYP2C9CYP2C19
SCHEMBL6974475 0.90 CYP1A2 (0.45) SMN1; SMN2TSHRATMCYP2C9CYP2C19
SCHEMBL7081165 0.89 LMNA (0.35) SMN1; SMN2TSHRATMCYP2C9CYP2C19
SCHEMBL6974432 0.88 EPHX1 (0.35) SMN1; SMN2CYP2C9CYP2C19CYP1A2EPHX1
SCHEMBL6972949 0.88 ALOX12 (0.37) SMN1; SMN2TP53
SCHEMBL6968991 0.87 LMNA (0.41) TSHRATMCYP2C9CYP2C19CYP1A2
SCHEMBL7087523 0.87 TOP2A (0.44) SMN1; SMN2TSHRATMCYP2C9CYP2C19
SCHEMBL6969941 0.86 CYP1A2 (0.39) SMN1; SMN2CYP2C9CYP2C19CYP1A2MEN1
SCHEMBL6969825 0.86 LMNA (0.31) MAPTNPSR1
SCHEMBL6972373 0.86 PIM1 (0.36) SMN1; SMN2TSHRCYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed