SCHEMBL6965525

SCHEMBL6965525

Cc1cc(C)cc(Sc2c(C(C)C)nc(CCCO)n2Cc2ccncc2)c1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.34
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TLR7 Q9NYK1 2/20 0.32
KCNH2 Q12809 1/20 0.31
ENPP2 Q13822 1/20 0.31
P2RX3 P56373 1/20 0.30
TSHR P16473 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972780 0.94 MEN1 (0.33) GSK3BMEN1KMT2AKCNH2ENPP2
SCHEMBL7081183 0.91 TDP1 (0.37) GSK3BALDH1A1TDP1TLR7TSHR
SCHEMBL6966489 0.90 TLR8 (0.35) GSK3BALDH1A1TDP1TLR7KCNH2
SCHEMBL7083001 0.89 MEN1 (0.34) ALDH1A1MEN1KMT2AKCNH2P2RX3
SCHEMBL6969774 0.89 ENPP2 (0.35) GSK3BALDH1A1TDP1TLR7ENPP2
SCHEMBL7082316 0.88 TLR7 (0.36) ALDH1A1TDP1TLR7
SCHEMBL7086620 0.88 GSK3B (0.40) GSK3BALDH1A1TDP1TLR7
SCHEMBL7083480 0.85 TLR8 (0.37) GSK3BALDH1A1TDP1TLR7KCNH2
SCHEMBL6968648 0.85 P2RX3 (0.33) GSK3BALDH1A1MEN1KMT2ATLR7
SCHEMBL7085890 0.84 GSK3B (0.34) GSK3BALDH1A1TDP1KMT2ATLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed