SCHEMBL7083480

SCHEMBL7083480

CC(C)c1nc(CCCO)n(Cc2ccncc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 3/20 0.37
GSK3B P49841 1/20 0.35
IDO1 P14902 1/20 0.34
ALDH1A1 P00352 3/20 0.34
TDP1 Q9NUW8 3/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
THRB P10828 1/20 0.33
TLR7 Q9NYK1 2/20 0.32
KCNH2 Q12809 2/20 0.32
TRPC4 Q9UBN4 1/20 0.32
TRPC5 Q9UL62 1/20 0.32
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959029 0.94 IDO1 (0.35) GSK3BIDO1ALDH1A1TDP1KDM4E
SCHEMBL6966489 0.91 TLR8 (0.35) TLR8GSK3BALDH1A1TDP1TLR7
SCHEMBL7084751 0.91 ALDH1A1 (0.38) TLR8ALDH1A1TDP1KDM4ELMNA
SCHEMBL7079909 0.90 IDO1 (0.36) IDO1ALDH1A1TDP1KDM4EHPGD
SCHEMBL7085890 0.90 GSK3B (0.34) GSK3BALDH1A1TDP1LMNATLR7
SCHEMBL7086620 0.89 GSK3B (0.40) GSK3BALDH1A1TDP1KDM4ETLR7
SCHEMBL6974232 0.88 IDO1 (0.35) GSK3BIDO1ALDH1A1TDP1KDM4E
SCHEMBL6971946 0.87 TLR8 (0.40) TLR8ALDH1A1TDP1KDM4ELMNA
SCHEMBL6967782 0.87 LMNA (0.39) IDO1ALDH1A1TDP1KDM4ELMNA
SCHEMBL6967360 0.86 IDO1 (0.36) IDO1ALDH1A1TDP1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed