SCHEMBL6965644

SCHEMBL6965644

COc1ccc2c(c1)CN(C(=O)c1ccc([N+](=O)[O-])cc1)c1ccccc1C2=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
ACHE P22303 1/20 0.44
BACE1 P56817 1/20 0.44
RAB9A P51151 1/20 0.44
MAPT P10636 5/20 0.43
LMNA P02545 1/20 0.43
ALDH1A1 P00352 3/20 0.43
TSHR P16473 1/20 0.43
KDM4E B2RXH2 1/20 0.42
KCNN4 O15554 1/20 0.42
KCNA3 P22001 1/20 0.42
MEN1 O00255 1/20 0.41
AHR P35869 1/20 0.41
KMT2A Q03164 1/20 0.41
HPGD P15428 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970953 0.85 RAB9A (0.47) SMN1; SMN2ACHEBACE1RAB9AMAPT
SCHEMBL7330482 0.78 HPGD (0.54) SMN1; SMN2RAB9AMAPTLMNAALDH1A1
SCHEMBL8961720 0.75 AVPR2 (0.51)
SCHEMBL3044124 0.75 KCNN4 (0.68) SMN1; SMN2MAPTALDH1A1KCNN4KCNA3
SCHEMBL7344427 0.74 CA1 (0.54) SMN1; SMN2MAPTLMNAALDH1A1TSHR
SCHEMBL7344362 0.74 CA1 (0.71) SMN1; SMN2RAB9AMAPTLMNAALDH1A1
SCHEMBL14509691 0.72 PTPN11 (0.42) MAPTLMNAALDH1A1KDM4EMEN1
SCHEMBL7353072 0.72 TSHR (0.61) SMN1; SMN2RAB9AMAPTLMNAALDH1A1
SCHEMBL7352575 0.70 ALDH1A1 (0.56) RAB9AMAPTLMNAALDH1A1TSHR
SCHEMBL4251148 0.70 NPC1 (0.58) SMN1; SMN2RAB9AMAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed