SCHEMBL6965840

SCHEMBL6965840

CCn1ncc(-c2ccc3c(ccn3-c3ccc(F)cc3)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.48
HTR1A P08908 2/20 0.45
HTR1B P28222 2/20 0.45
NR3C1 P04150 9/20 0.39
PGR P06401 5/20 0.38
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
ALOX12 P18054 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
DRD2 P14416 1/20 0.36
MCHR1 Q99705 1/20 0.35
EPHX2 P34913 1/20 0.35
SCN9A Q15858 1/20 0.35
CACNA1H O95180 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967960 0.85 KCNH2 (0.50) KCNH2HTR1AHTR1BNR3C1PGR
SCHEMBL6964471 0.79 DRD2 (0.54) KCNH2HTR1AHTR1BNR3C1PGR
SCHEMBL6969011 0.79 KCNH2 (0.48) KCNH2KDM4ENPC1ALDH1A1MAPT
SCHEMBL6957190 0.78 KCNH2 (0.47) KCNH2HTR1AHTR1BNR3C1KDM4E
SCHEMBL6967276 0.74 DRD2 (0.55) KCNH2HTR1AHTR1BNR3C1PGR
SCHEMBL6966566 0.73 KCNH2 (0.50) KCNH2HTR1AHTR1BKDM4ENPC1
SCHEMBL6966311 0.73 KCNH2 (0.52) KCNH2HTR1AHTR1BNR3C1PGR
SCHEMBL6960921 0.73 KCNH2 (0.49) KCNH2NR3C1KDM4ENPC1ALDH1A1
SCHEMBL6960229 0.72 DRD2 (0.54) KCNH2HTR1AHTR1BKDM4ENPC1
SCHEMBL6375040 0.72 KCNH2 (0.48) KCNH2NR3C1PGRKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602889-B1 5-heteroaryl substituted indoles H. LUNDBECK A.S. (DK) 2003-08-05 US disclosed
EP-1068198-B1 5-HETEROARYL SUBSTITUTED INDOLES LUNDBECK & CO AS H (DK) 2003-05-28 EP disclosed