SCHEMBL6966537

SCHEMBL6966537

CC(=O)NCc1nc(C(C)C)c(Sc2cccc(F)c2)n1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MTNR1A P48039 3/20 0.35
MTNR1B P49286 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
GAA P10253 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PIK3CA P42336 1/20 0.35
NOTUM Q6P988 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SLC6A9 P48067 2/20 0.34
POLB P06746 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973934 0.91 EPHX1 (0.37) NPSR1MAOAMAOBCA2CA4
SCHEMBL6961581 0.89 SMN1; SMN2 (0.32) NPSR1SMN1; SMN2L3MBTL1
SCHEMBL7084176 0.88 SMN1; SMN2 (0.38) NPSR1CA2CA4MTNR1AMTNR1B
SCHEMBL6974325 0.87 TP53 (0.39) NPSR1MAOAMAOBMTNR1AMTNR1B
SCHEMBL6961492 0.87 MAOA (0.36) NPSR1MAOAMAOBCA2CA4
SCHEMBL7084094 0.87 SMN1; SMN2 (0.40) NPSR1MTNR1AMTNR1BCYP1A2CYP2C9
SCHEMBL7087555 0.84 GCGR (0.38) NPSR1MAOAMAOBCYP1A2CYP3A4
SCHEMBL6967331 0.84 MAOA (0.36) NPSR1MAOAMAOBCA2CA4
SCHEMBL6962728 0.84 CYP1A2 (0.40) NPSR1MAOAMAOBCA2CA4
SCHEMBL6972012 0.84 RAB9A (0.41) GAACYP2D6CYP2C9CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed