SCHEMBL7084094

SCHEMBL7084094

CC(=O)NCc1nc(C(C)C)c(Sc2ccccc2)n1C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.40
MTNR1A P48039 7/20 0.39
MTNR1B P49286 7/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
NPSR1 Q6W5P4 1/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
ELANE P08246 1/20 0.36
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
POLB P06746 1/20 0.35
SETDB1 Q15047 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084970 0.89 MAPT (0.37) SMN1; SMN2MAPTMEN1CYP1A2CYP2C9
SCHEMBL6974325 0.87 TP53 (0.39) MTNR1AMTNR1BL3MBTL1NPSR1MAPT
SCHEMBL6966537 0.87 NPSR1 (0.36) SMN1; SMN2MTNR1AMTNR1BL3MBTL1NPSR1
SCHEMBL7084307 0.86 SMN1; SMN2 (0.44) SMN1; SMN2MTNR1AMTNR1BL3MBTL1NPSR1
SCHEMBL6974787 0.85 SMN1; SMN2 (0.35) SMN1; SMN2MAPTKDM4ENPC1RAB9A
SCHEMBL6965470 0.83 SETDB1 (0.33) SMN1; SMN2L3MBTL1NPSR1POLBSETDB1
SCHEMBL6961581 0.83 SMN1; SMN2 (0.32) SMN1; SMN2L3MBTL1NPSR1MAPTNPC1
SCHEMBL6972012 0.83 RAB9A (0.41) SMN1; SMN2L3MBTL1MAPTMEN1CYP2C9
SCHEMBL6966247 0.82 CYP1A2 (0.49) SMN1; SMN2L3MBTL1MAPTMEN1CYP1A2
SCHEMBL6970053 0.82 PTPN1 (0.34) SMN1; SMN2MAPTKDM4EPOLBSETDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed