SCHEMBL6973934

SCHEMBL6973934

CC(C)c1nc(CNC(N)=O)n(C)c1Sc1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.37
CA2 P00918 2/20 0.37
CA4 P22748 2/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
HDAC6 Q9UBN7 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
GAA P10253 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NOTUM Q6P988 1/20 0.34
TYMS P04818 1/20 0.34
SLC6A9 P48067 3/20 0.33
POLB P06746 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966537 0.91 NPSR1 (0.36) EPHX1CA2CA4MAOAMAOB
SCHEMBL6965334 0.89 PARP1 (0.30)
SCHEMBL6968447 0.88 CA2 (0.38) EPHX1CA2CA4CYP1A2CYP3A4
SCHEMBL6971356 0.88 TP53 (0.38) MAOAMAOBNPSR1TYMSPOLB
SCHEMBL7084970 0.87 MAPT (0.37) EPHX1CYP1A2CYP3A4GAACYP2C9
SCHEMBL6961492 0.86 MAOA (0.36) CA2CA4MAOAMAOBHDAC6
SCHEMBL6969795 0.84 EPHX1 (0.37) EPHX1CA2CA4MAOAMAOB
SCHEMBL7079210 0.84 LMNA (0.37) GAACYP2D6CYP2C9CYP2C19POLB
SCHEMBL6973797 0.83 MAOA (0.38) EPHX1CA2CA4MAOAMAOB
SCHEMBL7087555 0.83 GCGR (0.38) EPHX1MAOAMAOBCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed