SCHEMBL6966562

SCHEMBL6966562

Nc1ccc(NC(=O)CN(Cc2ccccc2)C(=O)C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
LMNA P02545 1/20 0.45
ACHE P22303 2/20 0.44
BCHE P06276 1/20 0.44
MTOR P42345 1/20 0.43
CYP3A4 P08684 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
CALCRL Q16602 2/20 0.43
KDM4E B2RXH2 2/20 0.43
MAP2K2 P36507 1/20 0.43
ADM2 Q7Z4H4 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MAPT P10636 1/20 0.41
LTA4H P09960 1/20 0.41
MLYCD O95822 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955771 0.83 MMP1 (0.54) ALDH1A1LMNAACHEMAPT
SCHEMBL6968790 0.82 KDM4E (0.47) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL6956260 0.76 RCE1 (0.49) KDM4EMLYCD
SCHEMBL6967760 0.76 RCE1 (0.49) KDM4EMLYCD
SCHEMBL16373478 0.76 CES1 (0.52) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL2413298 0.74 HDAC1 (0.59) CYP3A4
SCHEMBL6956921 0.73 GRIN2D (0.45) ALDH1A1NPSR1CYP2C19LMNAKDM4E
SCHEMBL3453783 0.72 EPHX2 (0.76) ALDH1A1LMNAACHEBCHEKDM4E
SCHEMBL7472989 0.71 ALDH1A1 (0.62) ALDH1A1NPSR1LMNAACHEBCHE
SCHEMBL16366240 0.71 GYS1 (0.39) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed