SCHEMBL6955771

SCHEMBL6955771

O=C(CN(Cc1ccccc1)C(=O)C(F)(F)F)Nc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 6/20 0.54
MMP2 P08253 6/20 0.54
MMP9 P14780 6/20 0.54
MMP8 P22894 6/20 0.54
MMP13 P45452 6/20 0.54
CRHBP P24387 1/20 0.53
CRHR2 Q13324 1/20 0.53
MAPT P10636 4/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
LMNA P02545 2/20 0.47
ALDH1A1 P00352 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HTT P42858 2/20 0.47
HSP90AA1 P07900 1/20 0.46
MAPK1 P28482 1/20 0.46
POLB P06746 2/20 0.46
NPC1 O15118 1/20 0.46
MITF O75030 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4194549 0.85 MMP1 (0.67) MMP1MMP2MMP9MMP8MMP13
SCHEMBL6957148 0.84 CRHBP (0.65) MMP1MMP2MMP9MMP8MMP13
SCHEMBL6966562 0.83 ALDH1A1 (0.47) MAPTLMNAALDH1A1ACHE
SCHEMBL11143290 0.79 ALDH1A1 (0.69) MMP1MMP2MMP9MMP8MMP13
SCHEMBL6957942 0.79 KCNH2 (0.64) MMP1MMP2MMP9MMP8MMP13
SCHEMBL6962369 0.79 KCNH2 (0.64) MMP1MMP2MMP9MMP8MMP13
SCHEMBL5179973 0.78 MMP1 (0.58) MMP1MMP2MMP9MMP8MMP13
SCHEMBL6963390 0.76 ALDH1A1 (0.59) CRHBPCRHR2MAPTMEN1KMT2A
SCHEMBL27841700 0.75 MEN1 (0.74) MAPTMEN1KMT2ALMNAALDH1A1
SCHEMBL16366561 0.74 ALDH1A1 (0.50) CRHBPCRHR2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed