SCHEMBL6966716

SCHEMBL6966716

CCn1c(COC(N)=O)nc(Sc2cc(C)cc(C)c2)c1C(C)C

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.32
NPC1 O15118 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079152 0.90 NPC1 (0.32) RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL6973926 0.88 LMNA (0.30) LMNA
SCHEMBL6968519 0.88 CYP1A2 (0.34) L3MBTL1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6969923 0.87 LMNA (0.36) RAB9ANPC1SMN1; SMN2L3MBTL1CYP1A2
SCHEMBL6972661 0.86 POLB (0.37) SMN1; SMN2L3MBTL1LMNA
SCHEMBL6971287 0.86 ALDH1A1 (0.36) RAB9ANPC1SMN1; SMN2L3MBTL1CYP1A2
SCHEMBL8113749 0.85 MEN1 (0.34) RAB9ANPC1SMN1; SMN2
SCHEMBL6969825 0.83 LMNA (0.31) LMNAMAPTNPSR1
SCHEMBL6965465 0.83 ALOX12 (0.41) RAB9ASMN1; SMN2L3MBTL1CYP1A2CYP3A4
SCHEMBL7081810 0.83 CA2 (0.38) SMN1; SMN2L3MBTL1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed