SCHEMBL6968937

SCHEMBL6968937

CNC(=S)OCc1nc(C(C)C)c(Sc2ccccc2)n1Cc1ccncc1

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.32
TP53 P04637 1/20 0.32
P2RX3 P56373 2/20 0.31
ALDH1A1 P00352 1/20 0.31
TOP2A P11388 1/20 0.31
TOP2B Q02880 1/20 0.31
ENPP2 Q13822 1/20 0.30
POLB P06746 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ITGB2 P05107 1/20 0.30
ICAM1 P05362 1/20 0.30
ITGAL P20701 1/20 0.30
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961267 0.90 ALDH1A1 (0.34) MAPTTP53P2RX3ALDH1A1
SCHEMBL6976430 0.90 HTT (0.34) ALDH1A1TLR7
SCHEMBL6967842 0.89 ENPP2 (0.33) TP53P2RX3ENPP2
SCHEMBL6961663 0.89 P2RX3 (0.31) P2RX3
SCHEMBL6974505 0.89 TOP2A (0.42) P2RX3ALDH1A1TOP2ATOP2BENPP2
SCHEMBL7083670 0.88 ENPP2 (0.33) P2RX3ENPP2
SCHEMBL6963992 0.86 MAPT (0.37) MAPTALDH1A1POLB
SCHEMBL6975076 0.86 TOP2A (0.31) ALDH1A1TOP2ATOP2B
SCHEMBL7182670 0.86 TLR7 (0.31) TP53ALDH1A1POLBKDM4ETLR7
SCHEMBL6975053 0.85 MEN1 (0.41) MAPTTP53P2RX3ALDH1A1ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed