SCHEMBL6976430

SCHEMBL6976430

CNC(=S)OCc1nc(C(C)C)c(Sc2ccccc2)n1Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
S1PR3 Q99500 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
ALOX5AP P20292 1/20 0.33
CYP3A4 P08684 1/20 0.33
HIF1A Q16665 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
KEAP1 Q14145 1/20 0.32
BLM P54132 1/20 0.32
SRC P12931 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085898 0.90 ALDH1A1 (0.37) HTTSMN1; SMN2S1PR3ALDH1A1GAA
SCHEMBL7083490 0.90 GRIN1 (0.35) HTTSMN1; SMN2S1PR3TLR7CYP3A4
SCHEMBL6968937 0.90 MAPT (0.32) TLR7ALDH1A1
SCHEMBL6974277 0.90 GRIN1 (0.34) HTTSMN1; SMN2S1PR3TLR7ALDH1A1
SCHEMBL7080182 0.90 MAPT (0.35) HTTSMN1; SMN2S1PR3HIF1AALDH1A1
SCHEMBL6964229 0.89 TOP2A (0.41) S1PR3CYP3A4
SCHEMBL6962639 0.87 RXFP1 (0.37) HTTSMN1; SMN2ALDH1A1GAA
SCHEMBL6969306 0.86 KMT2A (0.39) HTTSMN1; SMN2S1PR3CYP3A4HIF1A
SCHEMBL7086385 0.85 TLR7 (0.35) HTTS1PR3TLR7CYP3A4HIF1A
SCHEMBL6975076 0.84 TOP2A (0.31) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed