SCHEMBL6969044

SCHEMBL6969044

CCn1c(C)nc2cc(Sc3cccc4cnccc34)c([N+](=O)[O-])cc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
RAD52 P43351 1/20 0.36
KMT2A Q03164 4/20 0.36
TDP1 Q9NUW8 4/20 0.36
MEN1 O00255 3/20 0.36
MAPT P10636 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
GAA P10253 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 3/20 0.35
RAB9A P51151 2/20 0.35
PSMD14 O00487 1/20 0.35
ALDH1A1 P00352 3/20 0.35
LMNA P02545 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
CYP1A2 P05177 1/20 0.34
HASPIN Q8TF76 2/20 0.33
TSHR P16473 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963410 0.96 KDM4E (0.36) KDM4ERAD52KMT2ATDP1MEN1
SCHEMBL6974563 0.81 KDM4E (0.41) KDM4ERAD52KMT2ATDP1MAPT
SCHEMBL6971485 0.80 LMNA (0.40) KMT2AMEN1GAAL3MBTL1MAPK1
SCHEMBL6973974 0.79 LMNA (0.40) KMT2AMEN1GAAL3MBTL1MAPK1
SCHEMBL6970234 0.78 MAPT (0.46) KDM4EKMT2ATDP1MEN1MAPT
SCHEMBL6974578 0.77 HTT (0.41) KMT2ATDP1MEN1MAPTNPSR1
SCHEMBL8357964 0.76 SLC6A2 (0.49) KDM4EKMT2ATDP1MEN1MAPT
SCHEMBL6971375 0.76 MAPT (0.44) KDM4EKMT2ATDP1MEN1MAPT
SCHEMBL6963335 0.75 LMNA (0.46) KMT2ATDP1MEN1MAPTNPSR1
SCHEMBL6972315 0.75 LMNA (0.46) KMT2ATDP1MEN1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed