SCHEMBL6971375

SCHEMBL6971375

Cc1nc2cc(Sc3cccc4cnccc34)c([N+](=O)[O-])cc2c(=O)[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.44
GAA P10253 2/20 0.44
RAB9A P51151 2/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 1/20 0.44
USP2 O75604 1/20 0.44
GLA P06280 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TYMS P04818 2/20 0.43
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
NPSR1 Q6W5P4 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CDC7 O00311 1/20 0.38
DBF4 Q9UBU7 1/20 0.38
HTT P42858 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970234 0.81 MAPT (0.46) MAPTGAARAB9AALDH1A1KDM4E
SCHEMBL6961855 0.80 MEN1 (0.41) MAPTGAARAB9AALDH1A1HPGD
SCHEMBL6967350 0.79 SMN1; SMN2 (0.44) MAPTGAARAB9AALDH1A1KDM4E
SCHEMBL6974578 0.79 HTT (0.41) MAPTGAARAB9AALDH1A1NPC1
SCHEMBL8357964 0.79 SLC6A2 (0.49) MAPTGAARAB9AALDH1A1KDM4E
SCHEMBL6963335 0.77 LMNA (0.46) MAPTGAARAB9AALDH1A1SMN1; SMN2
SCHEMBL6972315 0.77 LMNA (0.46) MAPTGAARAB9AALDH1A1SMN1; SMN2
SCHEMBL6970313 0.76 PGR (0.39) MAPTGAARAB9AALDH1A1NPC1
SCHEMBL6974324 0.76 KMT2A (0.40) MAPTGAARAB9AALDH1A1HPGD
SCHEMBL6959978 0.76 KMT2A (0.40) MAPTGAARAB9AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed