SCHEMBL6974563

SCHEMBL6974563

CCn1c(C)nc2cc(Cl)c(Sc3cccc4cnccc34)cc21

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
RAD52 P43351 1/20 0.39
DCTPP1 Q9H773 2/20 0.38
KMT2A Q03164 2/20 0.37
TSHR P16473 2/20 0.37
MAPT P10636 2/20 0.37
TDP1 Q9NUW8 1/20 0.36
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
RHEB Q15382 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963410 0.83 KDM4E (0.36) KDM4ERAD52KMT2ATSHRMAPT
SCHEMBL6969044 0.81 KDM4E (0.36) KDM4ERAD52KMT2ATSHRMAPT
SCHEMBL6962804 0.76 TNF (0.47) DCTPP1CYP11B2RAB9A
SCHEMBL1048487 0.72 KDM4E (0.58) KDM4ERAD52DCTPP1KMT2ATSHR
SCHEMBL6962927 0.72 LMNA (0.51) KDM4ERAD52MAPTLMNASMN1; SMN2
SCHEMBL6968741 0.71 KDM4E (0.57) KDM4EKMT2AMAPTLMNASMN1; SMN2
SCHEMBL6963124 0.70 LMNA (0.41) KDM4EMAPTLMNASMN1; SMN2ALDH1A1
SCHEMBL6973974 0.67 LMNA (0.40) KMT2ATSHRLMNASMN1; SMN2RAB9A
SCHEMBL6971485 0.67 LMNA (0.40) KMT2ATSHRLMNASMN1; SMN2RAB9A
SCHEMBL6963171 0.66 AR (0.53) KDM4ELMNACYP11B1CYP11B2RHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed