SCHEMBL6970858

SCHEMBL6970858

OC1(c2ccc3[nH]cc(CCN4CCCC4)c3c2)C=CSC=C1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MPO P05164 3/20 0.58
HTR1D P28221 10/20 0.56
HTR1B P28222 10/20 0.56
HTR2A P28223 4/20 0.54
BRD4 O60885 1/20 0.47
HTR7 P34969 1/20 0.46
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969558 0.81 MPO (0.60) MPOHTR1DHTR1BHTR2ABRD4
SCHEMBL6967767 0.80 HTR1D (0.59) MPOHTR1DHTR1BHTR2ABRD4
SCHEMBL6966135 0.79 MPO (0.57) MPOHTR1DHTR1BHTR2ABRD4
SCHEMBL6965752 0.78 HTR1A (0.59) MPOHTR1DHTR1BHTR2AHTR7
SCHEMBL6967771 0.77 MPO (0.55) MPOHTR1DHTR1BHTR2ABRD4
SCHEMBL27095364 0.76 HTR7 (0.71) MPOHTR1DHTR1BHTR2AHTR7
SCHEMBL26989598 0.75 HTR7 (0.70) MPOHTR1DHTR1BHTR2AHTR7
SCHEMBL6968414 0.75 DRD3 (0.56) MPOHTR1DHTR1BHTR2AHTR2C
SCHEMBL8506914 0.74 HTR1D (0.71) MPOHTR1DHTR1BHTR2ABRD4
SCHEMBL733997 0.74 MPO (1.00) MPOHTR1DHTR1BHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1289479-C As 5-HT1D5-ring indole compounds of receptor ligands ALLELIX BIOPHARMA (CA) 2006-12-13 CN claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP claimed
CN-1245491-A 5-cyclo indole compounds as 5-HT receptor ligands ALLELIX BIOPHARMA (CA) 2000-02-23 CN claimed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US claimed
CN-1289479-C As 5-HT1D5-ring indole compounds of receptor ligands ALLELIX BIOPHARMA (CA) 2006-12-13 CN disclosed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
CN-1245491-A 5-cyclo indole compounds as 5-HT receptor ligands ALLELIX BIOPHARMA (CA) 2000-02-23 CN disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed