SCHEMBL6969917

SCHEMBL6969917

CC(C)c1nc(C=O)n(Cc2ccncc2)c1Sc1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
CYP3A4 P08684 5/20 0.34
CYP17A1 P05093 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
P2RX3 P56373 2/20 0.34
ATM Q13315 2/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
KMT2A Q03164 1/20 0.33
VDR P11473 1/20 0.32
CYP2D6 P10635 4/20 0.32
CYP2C9 P11712 3/20 0.32
CYP1A2 P05177 3/20 0.32
CYP2C19 P33261 3/20 0.32
USP2 O75604 2/20 0.32
IDO1 P14902 1/20 0.32
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972005 0.91 VDR (0.32) GRIN1GRIN2BKMT2AVDR
SCHEMBL6970262 0.89 GRIN1 (0.41) GRIN1GRIN2BCYP11B2IDO1
SCHEMBL6969927 0.89 IDO1 (0.38) P2RX3LMNATP53KMT2AVDR
SCHEMBL6973384 0.87 GRIN1 (0.36) GRIN1GRIN2BCYP3A4CYP17A1CYP11B1
SCHEMBL6973380 0.87 GRIN1 (0.36) GRIN1GRIN2BCYP3A4CYP17A1CYP11B1
SCHEMBL6964826 0.87 VDR (0.36) CYP3A4P2RX3LMNAKMT2AVDR
SCHEMBL6968637 0.85 DHODH (0.34) ATMLMNAKMT2AALDH1A1
SCHEMBL6966500 0.85 PDE4A (0.39) CYP3A4ATMLMNAKMT2ACYP2C9
SCHEMBL6967288 0.84 GRIN1 (0.40) GRIN1GRIN2BKMT2AKDM4E
SCHEMBL7082707 0.84 GRIN1 (0.38) GRIN1GRIN2BCYP3A4CYP17A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed