SCHEMBL6970262

SCHEMBL6970262

CC(C)c1nc(C=O)n(Cc2cccnc2)c1Sc1cccc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 16/20 0.41
GRIN2B Q13224 16/20 0.41
CYP11B2 P19099 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
IDO1 P14902 1/20 0.33
TBXA2R P21731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967171 0.92 GRIN1 (0.41) GRIN1GRIN2BTLR7IDO1
SCHEMBL6969917 0.89 GRIN1 (0.38) GRIN1GRIN2BCYP11B2IDO1
SCHEMBL6970594 0.89 ALDH1A1 (0.40) GRIN1GRIN2BIDO1
SCHEMBL6962674 0.88 ALOX5AP (0.37)
SCHEMBL6973265 0.88 GRIN1 (0.39) GRIN1GRIN2BCYP11B2
SCHEMBL6973263 0.88 GRIN1 (0.39) GRIN1GRIN2BCYP11B2
SCHEMBL6973483 0.85 MAPT (0.37) CYP11B2
SCHEMBL6968924 0.85 GABRA5 (0.37) GRIN1GRIN2B
SCHEMBL6974887 0.84 GRIN1 (0.39) GRIN1GRIN2BCYP11B2TLR7
SCHEMBL7083464 0.84 GRIN1 (0.39) GRIN1GRIN2BCYP11B2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed