SCHEMBL6967288

SCHEMBL6967288

CC(C)c1nc(C=O)n(Cc2ccccn2)c1Sc1cccc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 13/20 0.40
GRIN2B Q13224 13/20 0.40
S1PR3 Q99500 2/20 0.35
KDM4E B2RXH2 1/20 0.34
BRD4 O60885 1/20 0.33
NOX4 Q9NPH5 2/20 0.33
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960341 0.92 S1PR3 (0.35) GRIN1GRIN2BS1PR3KDM4EBRD4
SCHEMBL6973368 0.89 ALDH1A1 (0.34) KDM4EBRD4NOX4KMT2A
SCHEMBL6973903 0.89 GRIN1 (0.38) GRIN1GRIN2BKDM4EBRD4NOX4
SCHEMBL6969251 0.88 GRIN1 (0.38) GRIN1GRIN2BS1PR3NOX4KMT2A
SCHEMBL6969252 0.88 GRIN1 (0.38) GRIN1GRIN2BS1PR3NOX4KMT2A
SCHEMBL6973761 0.85 CFTR (0.44) S1PR3KDM4EKMT2A
SCHEMBL6973236 0.84 ALDH1A1 (0.35) GRIN1GRIN2BS1PR3BRD4NOX4
SCHEMBL6969917 0.84 GRIN1 (0.38) GRIN1GRIN2BKDM4EKMT2A
SCHEMBL6968637 0.84 DHODH (0.34) KMT2A
SCHEMBL6967980 0.83 GRIN1 (0.39) GRIN1GRIN2BS1PR3KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed