SCHEMBL6969927

SCHEMBL6969927

CC(C)c1nc(C=O)n(Cc2ccncc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.38
TDP1 Q9NUW8 2/20 0.37
PDE4D Q08499 1/20 0.34
PDE4B Q07343 1/20 0.34
VDR P11473 2/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
KCNH2 Q12809 1/20 0.33
TERT O14746 1/20 0.33
POLB P06746 1/20 0.33
KDM4E B2RXH2 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967722 0.91 TDP1 (0.34) IDO1TDP1VDRKCNH2MEN1
SCHEMBL6970594 0.90 ALDH1A1 (0.40) IDO1TDP1KDM4EKMT2ALMNA
SCHEMBL6969917 0.89 GRIN1 (0.38) IDO1TDP1VDRKDM4EKMT2A
SCHEMBL6964826 0.88 VDR (0.36) TDP1VDRKDM4ENPSR1MEN1
SCHEMBL6960641 0.87 IDO1 (0.36) IDO1TDP1PDE4DPDE4BCSNK2A2
SCHEMBL6960647 0.87 IDO1 (0.36) IDO1TDP1PDE4DPDE4BCSNK2A2
SCHEMBL6974042 0.86 TP53 (0.36) TDP1VDRTERTPOLBNPSR1
SCHEMBL6966500 0.85 PDE4A (0.39) TDP1PDE4DPDE4BPOLBKDM4E
SCHEMBL6973903 0.85 GRIN1 (0.38) TDP1VDRKDM4ENPSR1MEN1
SCHEMBL6965090 0.84 IDO1 (0.38) IDO1TDP1PDE4DPDE4BVDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed