SCHEMBL6970053

SCHEMBL6970053

CC(C)c1nc(CNS(C)(=O)=O)n(C)c1Sc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.34
CDC25A P30304 1/20 0.34
CDC25B P30305 1/20 0.34
SETDB1 Q15047 1/20 0.34
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
DHFR P00374 1/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
ALDH1A1 P00352 2/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
POLB P06746 2/20 0.32
HPGD P15428 2/20 0.32
TSHR P16473 1/20 0.32
RECQL P46063 1/20 0.32
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6968203 0.87 MAOB (0.36) HPGDMAOAMAOB
SCHEMBL6967331 0.87 MAOA (0.36) SMN1; SMN2ALDH1A1MAPTPOLBMAOA
SCHEMBL7084653 0.86 SETDB1 (0.33) PTPN1CDC25ACDC25BSETDB1PTGS1
SCHEMBL6961217 0.84 MALT1 (0.32)
SCHEMBL6967136 0.84 GAA (0.33)
SCHEMBL6974787 0.84 SMN1; SMN2 (0.35) PTPN1CDC25ACDC25BDHFRSMN1; SMN2
SCHEMBL6975564 0.83 PKM (0.37) PTGS2SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL7084094 0.82 SMN1; SMN2 (0.40) SETDB1SMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL7084970 0.81 MAPT (0.37) SMN1; SMN2MAPTRECQL
SCHEMBL6964165 0.81 POLB (0.38) PTGS1PTGS2SMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed