SCHEMBL7084653

SCHEMBL7084653

CCn1c(CNS(C)(=O)=O)nc(C(C)C)c1Sc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SETDB1 Q15047 1/20 0.33
PTPN1 P18031 1/20 0.33
CDC25A P30304 1/20 0.33
CDC25B P30305 1/20 0.33
DHFR P00374 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
POLB P06746 2/20 0.32
THRB P10828 1/20 0.32
TLR7 Q9NYK1 1/20 0.31
KDM4E B2RXH2 1/20 0.30
TSHR P16473 1/20 0.30
RECQL P46063 1/20 0.30
PER2 O15055 1/20 0.30
CRY1 Q16526 1/20 0.30
CRY2 Q49AN0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973826 0.87 ALDH1A1 (0.34) DHFRPER2CRY1CRY2
SCHEMBL6973819 0.87 TP53 (0.35) TSHR
SCHEMBL6970053 0.86 PTPN1 (0.34) SETDB1PTPN1CDC25ACDC25BDHFR
SCHEMBL6964165 0.85 POLB (0.38) PTGS1PTGS2POLBTHRBKDM4E
SCHEMBL7082939 0.84 SMN1; SMN2 (0.31) PTPN1CDC25ACDC25BDHFR
SCHEMBL6968974 0.84 ALDH1A1 (0.31)
SCHEMBL6974402 0.84 TDP1 (0.32)
SCHEMBL7077261 0.84 POLB (0.35) POLBTHRBTLR7
SCHEMBL7088075 0.84 MAPT (0.37) PTGS2
SCHEMBL7087408 0.83 POLB (0.38) PTGS1PTGS2POLBTHRBTLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed