SCHEMBL6970158

SCHEMBL6970158

O=[N+]([O-])c1ccc2[nH]nnc2c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.37
ATM Q13315 1/20 0.37
NOS1 P29475 4/20 0.35
CASP6 P55212 3/20 0.34
MAPT P10636 7/20 0.33
ALDH1A1 P00352 6/20 0.33
MEN1 O00255 5/20 0.33
KMT2A Q03164 5/20 0.33
KDM4E B2RXH2 4/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
LMNA P02545 3/20 0.33
BLM P54132 3/20 0.33
CYP3A4 P08684 3/20 0.33
TSHR P16473 3/20 0.33
IDO1 P14902 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 2/20 0.33
NOS2 P35228 2/20 0.33
POLB P06746 2/20 0.33
THRB P10828 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3728212 0.81 TSHR (0.37) TDP1NOS1CASP6MAPTALDH1A1
SCHEMBL32679425 0.81 TSHR (0.37) TDP1NOS1CASP6MAPTALDH1A1
SCHEMBL6052169 0.80 GPR35 (0.44) TDP1NOS1CASP6MAPTALDH1A1
SCHEMBL27647699 0.80 TDP1 (0.44) TDP1NOS1MAPTALDH1A1MEN1
SCHEMBL3730228 0.80 MAPT (0.40) TDP1NOS1CASP6MAPTALDH1A1
Silver SCHEMBL9168054 0.79 GPR35 (0.43) TDP1NOS1CASP6MAPTALDH1A1
SCHEMBL9168064 0.79 GPR35 (0.43) TDP1NOS1CASP6MAPTALDH1A1
SCHEMBL6052000 0.76 TDP1 (0.43) TDP1CASP6MAPTALDH1A1MEN1
SCHEMBL103130 0.76 NOS1 (0.51) TDP1NOS1MAPTALDH1A1MEN1
Silver SCHEMBL9169439 0.75 MAPT (0.33) TDP1NOS1CASP6MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed