SCHEMBL6970557

SCHEMBL6970557

CC(=O)OCCc1nc(C(C)C)c(Sc2cc(Cl)cc(Cl)c2)n1Cc1ccccn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HSP90AA1 P07900 1/20 0.33
HSP90B1 P14625 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TP53 P04637 1/20 0.32
SLC16A3 O15427 1/20 0.32
ADRA1D P25100 1/20 0.32
S1PR3 Q99500 5/20 0.32
P2RX3 P56373 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NPC1 O15118 1/20 0.32
HDAC1 Q13547 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087678 0.93 MEN1 (0.33) MEN1KMT2AHSP90AA1HSP90B1TAS1R3
SCHEMBL7084635 0.92 ADRA1D (0.35) MEN1KMT2AHSP90AA1HSP90B1TP53
SCHEMBL7078972 0.91 SLC16A3 (0.35) MEN1KMT2AHSP90AA1HSP90B1TP53
SCHEMBL6966916 0.90 CYP1A2 (0.35) MEN1KMT2ATAS1R3TAS1R1TP53
SCHEMBL6972647 0.87 ADRA1D (0.34) MEN1KMT2AHSP90AA1HSP90B1TP53
SCHEMBL8343030 0.87 LMNA (0.40) MEN1KMT2ATP53SLC16A3ADRA1D
SCHEMBL6974113 0.86 S1PR3 (0.38) KMT2AS1PR3
SCHEMBL7082531 0.86 HRH1 (0.34) MEN1KMT2AHSP90AA1HSP90B1TP53
SCHEMBL6973716 0.86 HSP90AA1 (0.36) MEN1KMT2AHSP90AA1HSP90B1TP53
SCHEMBL6973416 0.86 MAPT (0.36) KMT2ATP53SLC16A3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed