SCHEMBL6973716

SCHEMBL6973716

COC(=O)CCc1nc(C(C)C)c(Sc2cc(Cl)cc(Cl)c2)n1Cc1ccccn1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.36
HSP90B1 P14625 1/20 0.36
ENPP2 Q13822 8/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TP53 P04637 2/20 0.34
S1PR3 Q99500 2/20 0.33
MAPT P10636 2/20 0.33
P2RX3 P56373 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973417 0.93 MAPT (0.37) HSP90AA1HSP90B1ENPP2KDM4EALDH1A1
SCHEMBL8343030 0.90 LMNA (0.40) ENPP2MEN1KMT2ATP53
SCHEMBL6974458 0.90 S1PR3 (0.38) ENPP2KDM4EALDH1A1SMN1; SMN2HPGD
SCHEMBL7082531 0.86 HRH1 (0.34) HSP90AA1HSP90B1KDM4EALDH1A1MEN1
SCHEMBL6970557 0.86 MEN1 (0.34) HSP90AA1HSP90B1KDM4EALDH1A1SMN1; SMN2
SCHEMBL6968985 0.86 KDM4E (0.38) ENPP2KDM4EMAPTP2RX3
SCHEMBL7084635 0.85 ADRA1D (0.35) HSP90AA1HSP90B1KDM4EALDH1A1SMN1; SMN2
SCHEMBL6973437 0.85 MEN1 (0.40) ALDH1A1HPGDMEN1KMT2ATP53
SCHEMBL6970195 0.85 TLR7 (0.35) HSP90B1KDM4EALDH1A1MEN1KMT2A
SCHEMBL7082928 0.85 HRH1 (0.36) HSP90B1KDM4EALDH1A1S1PR3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed