SCHEMBL6970675

SCHEMBL6970675

O=C1CCCCC(CCC2CCCCN2)N1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
FDPS P14324 2/20 0.40
HRH3 Q9Y5N1 3/20 0.40
POLB P06746 1/20 0.39
FKBP5 Q13451 1/20 0.38
CRBN Q96SW2 1/20 0.38
CYP2D6 P10635 3/20 0.37
CYP1A2 P05177 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
MLNR O43193 1/20 0.37
ABCB11 O95342 1/20 0.37
EGFR P00533 1/20 0.37
FYN P06241 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
HTR1A P08908 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29742940 0.87 KMT2A (0.35) KMT2AFKBP5CRBNALDH1A1
SCHEMBL6977209 0.79 HRH3 (0.40) KMT2AFDPSHRH3POLBCYP2D6
SCHEMBL6444135 0.78 NOS1 (0.37) KMT2AALDH1A1OPRM1
SCHEMBL2989773 0.78 IRAK4 (0.32) FKBP5CRBN
SCHEMBL11025505 0.78 NOS3 (0.38) KMT2AFKBP5CRBNSIGMAR1
Hydrochloric Acid SCHEMBL6971032 0.77 KMT2A (0.40) KMT2AFDPSHRH3POLBCYP2D6
SCHEMBL4019894 0.77 CRBN (0.36) KMT2AFKBP5CRBNALDH1A1
SCHEMBL6971926 0.76 PDCD1 (0.30)
SCHEMBL1423906 0.75 ALDH1A1 (0.41) KMT2ACYP1A2MEN1ALDH1A1TP53
SCHEMBL6981344 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP disclosed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US disclosed
EP-0821674-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1998-02-04 EP disclosed
WO-1996033175-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1996-10-24 WO disclosed