SCHEMBL6970712

SCHEMBL6970712

NCCCCCCC(=O)N1CCC(c2nc(N)nc3ccccc23)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.45
TNKS O95271 12/20 0.45
PARP2 Q9UGN5 12/20 0.45
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 2/20 0.40
HPGD P15428 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CYP1A2 P05177 1/20 0.40
NUDT1 P36639 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981163 1.00 PARP1 (0.45) PARP1TNKSPARP2HSP90AA1HSP90AB1
SCHEMBL6977139 1.00 PARP1 (0.45) PARP1TNKSPARP2HSP90AA1HSP90AB1
SCHEMBL6979788 0.82 SIGMAR1 (0.49) SIGMAR1
SCHEMBL6980502 0.82 SIGMAR1 (0.49) SIGMAR1
SCHEMBL6968387 0.79 ALDH1A1 (0.51) PARP1HSP90AA1HSP90AB1ALDH1A1HSD17B10
SCHEMBL6976291 0.78 LMNA (0.55) HSP90AA1HSP90AB1ALDH1A1HSD17B10HPGD
SCHEMBL6979861 0.76 ROCK1 (0.42) PARP1TNKSPARP2HSP90AA1HSP90AB1
SCHEMBL6981315 0.76 MEN1 (0.58) ALDH1A1
SCHEMBL6976998 0.76 KDM4E (0.53) ALDH1A1HSD17B10HPGDKDM4ECASP1
SCHEMBL6974607 0.76 NAMPT (0.50) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892795-B1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMA (JP) 2003-01-08 EP disclosed
EP-0892795-A1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1999-01-27 EP disclosed
WO-1997038992-A1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-10-23 WO disclosed